UK Clinical Pharmacy Association

Lurasidone

Issues for surgery

Risk of withdrawal if omitted (see Further information).

Risk of relapse of schizophrenia or bipolar disorder if omitted.

Advice in the perioperative period

Elective and emergency surgery

Continue.

Post-operative advice

If a long Nil by Mouth (NBM) period is anticipated, or if there are concerns regarding enteral absorption, advice on alternative preparations/routes should be sought from a psychiatrist.

If treatment with lurasidone (at doses >111mg) is interrupted for >3 days, consult product literature for advice on restarting.

Interactions with common anaesthetic agents

Central Nervous System (CNS) depression 

Also see Interactions with other common medicines used in the perioperative period.

Lurasidone has CNS depressant effects which may be additive with other medicines that also have CNS depressant effects such as:

  • benzodiazepines
  • inhalational anaesthetics and intravenous anaesthetics
  • local anaesthetics
  • opioids

Consult British National Formulary for available drugs in each class.

Hypotension

Lurasidone can increase the risk of hypotension when used concomitantly with inhalational and intravenous anaesthetics.

Interactions with other common medicines used in the perioperative period

CNS Depression 

Also see Interactions with common anaesthetic agents for information on opioids.

Lurasidone has CNS depressant effects which may be additive with antiemetics that also have CNS depressant effects, such as cyclizine, droperidol and prochlorperazine.

Hypotension

Lurasidone can increase the risk of hypotension when used concomitantly with droperidol and prochlorperazine.

Hypokalaemia

Dexamethasone and hydrocortisone may cause hypokalaemia (potentially increasing the risk of torsades de pointes) with amisulpride, paliperidone or risperidone – use with caution. If hypokalaemia occurs, corrective action should be taken and QT-interval monitored.

Antimicrobials

Macrolides

Clarithromycin is predicted to increase the exposure to lurasidone through inhibition of CYP3A4.

Myelosuppression

Concomitant use of lurasidone with the following can increase the risk of myelosuppression:

  • co-trimoxazole
  • linezolid
  • trimethoprim

Whilst single surgical prophylactic doses should not pose a problem, monitor for side effects and consider reducing lurasidone dose if a prolonged course of clarithromycin or ciprofloxacin is required, and monitor full blood count if a prolonged course of myelosuppressive medication is required.

Further information

Withdrawal

Abrupt withdrawal of lurasidone may result in symptoms including sweating, insomnia, tremor, anxiety, nausea and vomiting.

Venous thromboembolism (VTE)

Cases of VTE have been reported with antipsychotic drugs, although a causal relationship has not been established. Patients with schizophrenia often have acquired risk factors for VTE; identify any risk factors and consider if thromboprophylaxis is indicated post-operatively.

References

Baxter K, Preston CL (eds), Stockley’s Drug Interactions (online) London: Pharmaceutical Press. http://www.medicinescomplete.com [Accessed on 20th August 2019]

Joint Formulary Committee. British National Formulary (online) London: BMJ Group and Pharmaceutical Press. http://www.medicinescomplete.com [Accessed on 20th August 2019]

Summary of Product Characteristics – Latuda® (lurasidone) 18.5mg film-coated tablets. Sunovion Pharmaceuticals Europe Ltd. Accessed via www.medicines.org.uk 20/08/2019 [date of revision of the text December 2018]